942591-66-4Relevant academic research and scientific papers
Novel cyclic-imide peptidomimetics as aminopeptidase N inhibitors. Design, chemistry and activity evaluation. Part I
Li, Qianbin,Fang, Hao,Wang, Xuejian,Hu, Liping,Xu, Wenfang
experimental part, p. 4819 - 4825 (2010/02/27)
A series of aminopeptidase inhibitors with cyclic-imide scaffold are described. The biological characterization for the piperidinedione analogues revealed that most compounds displayed high inhibitory activity against APN. Among which 4l and 6 showed pote
