943240-83-3Relevant academic research and scientific papers
Design, synthesis, and structure-affinity relationship studies in NK1 receptor ligands based on azole-fused quinolinecarboxamide moieties
Cappelli, Andrea,Giuliani, Germano,Anzini, Maurizio,Riitano, Daniela,Giorgi, Gianluca,Vomero, Salvatore
, p. 6850 - 6859 (2008/12/21)
The substituent in position 2 of the quinoline nucleus of NK1 receptor ligands 5 has been constrained into different five-membered heterocyclic moieties in order to obtain information on the binding site pocket interacting with this apparently
HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS
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Page/Page column 10; 18-19, (2010/11/27)
The present invention relates to compounds of formula 1, method of preparation and uses thereof.
Condensed heterocyclic compounds, their production and use
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, (2008/06/13)
Novel compound represented by the formula: STR1 such as 6-Chloro-N-(2,6-diethoxyphenyl)-4-(2-methylphenyl-2-oxo-2H-1-benzopyran-3-acetamide: STR2 or a salt thereof. The compound has an excellent activity of inhibiting ACAT, lowering the cholesterol in blood and inhibiting tachykinin receptor. The present invention also relates to the production and use of the disclosed compound.
