943448-26-8Relevant articles and documents
The discovery of high affinity agonists of GPR109a with reduced serum shift and improved ADME properties
Imbriglio, Jason E.,Dirocco, Daniel,Bodner, Rena,Raghavan, Subharekha,Chen, Weichun,Marley, Daria,Esser, Craig,Holt, Tom G.,Wolff, Michael S.,Taggart, Andrew K.P.,Waters, M. Gerard,Tata, James R.,Colletti, Steven L.
, p. 2721 - 2724 (2011)
Amino-anthranilic acid derivatives have been identified as a new class of low serum shifted, high affinity full agonists of the human orphan G-protein-coupled receptor GPR109a with improved ADME properties.