943593-60-0

Upstream product

• 119090-32-3 N-(4-bromophenyl)-N-benzylhydrazine 
• 76782-82-6 tert-Butyldimethyl(prop-2-ynyloxy)silane 

Downstream Products

• 1007893-44-8 1-benzyl-3-(tert-butyldimethylsiloxy)-5-(2,6-dimethylphenoxy)-2-methyl-1H-indole 
• 1007893-48-2 4-[1-benzyl-3-(tert-butyldimethylsiloxy)-2-methyl-1H-indol-5-yl]naphthalen-1-ol 
• 1007893-45-9 1-benzyl-3-(tert-butyldimethylsiloxy)-5-(2-tert-butyl-4-methylphenoxy)-2-methyl-1H-indole 
• 1007893-40-4 1-benzyl-3-(tert-butyldimethylsiloxy)-2-methyl-5-(2-methylphenoxy)-1H-indole 
• 1034385-14-2 1-benzyl-5-bromo-2-methyl-3-(2-N,N-diethylaminoethoxy)indole 

Relevant academic research and scientific papers

Synthesis of 3-(2-N,N-diethylaminoethoxy)indoles as potential 5-HT 6 receptor ligands

The synthesis of new pharmaceutically interesting 3-(2-N,N- diethylaminoethoxy)indole derivatives is described. Starting from 3-silyloxy-2-methylindoles, deprotection and in situ aminoalkylation provided 3-(2-N,N-diethylaminoethoxy)indoles in good yield.

Titanium-catalyzed hydroamination of propargyl alcohol derivatives: Synthesis of 3-silyloxy-2-methylindoles via hydrohydrazination

A general method for the one-pot synthesis of substituted 3-(tert-butyldimethylsilyloxy)indoles via hydrohydrazination of alkynes and subsequent Fischer indole synthesis has been developed. For the first time titanium-catalyzed hydroaminations of propargy