944247-24-9Relevant academic research and scientific papers
Identification and SAR of potent and selective non-peptide obeline somatostatin sst1 receptor antagonists
Troxler, Thomas,Hoyer, Daniel,Langenegger, Daniel,Neumann, Peter,Pfaeffli, Paul,Schoeffter, Philippe,Sorg, Dieter,Swoboda, Robert,Hurth, Konstanze
, p. 3983 - 3987 (2008/02/13)
A novel class of non-peptide somatostatin receptor ligands bearing the octahydrobenzo[g]quinoline (obeline) structural element has been identified. SAR studies have been performed that led to the discovery of derivatives with high affinity (pKd
