947407-75-2Relevant articles and documents
Identification and optimization of novel 1,3,4-oxadiazole EP1 receptor antagonists
Hall, Adrian,Brown, Susan H.,Chowdhury, Anita,Giblin, Gerard M.P.,Gibson, Mairi,Healy, Mark P.,Livermore, David G.,McArthur Wilson, Richard J.,Naylor, Alan,Rawlings, D. Anthony,Roman, Shilina,Ward, Emma,Willay, Caroline
, p. 4450 - 4455 (2008/02/10)
A novel series of oxadiazole EP1 receptor antagonists was identified by replacing the amide of a known glycine sulfonamide derivative with a 1,3,4-oxadiazole. Optimization of the substitution patterns on the three aromatic rings led to the iden
