948993-91-7Relevant academic research and scientific papers
Identification of ortho-amino benzamides and nicotinamides as MCHr1 antagonists
Vasudevan, Anil,LaMarche, Matthew J.,Blackburn, Christopher,Che, Jennifer Lee,Luchaco-Cullis, Courtney A.,Lai, Sujen,Marsilje, Thomas H.,Patane, Michael A.,Souers, Andrew J.,Wodka, Derek,Geddes, Bradley,Chen, Sumiao,Brodjian, Seven,Falls, Doug H.,Dayton, Brian D.,Bush, Eugene,Brune, Michael,Shapiro, Robin D.,Marsh, Kennan C.,Hernandez, Lisa E.,Sham, Hing L.,Collins, Christine A.,Kym, Philip R.
, p. 4174 - 4179 (2005)
Several potent and efficacious MCHr1 antagonists containing an ortho-amino benzamide or nicotinamide chemotype have been identified, exemplified by 28 and 50.
