949100-76-9Relevant academic research and scientific papers
Discovery of novel free fatty acid receptor 1 agonists bearing triazole core via click chemistry
Li, Zheng,Yang, Jianyong,Wang, Xuekun,Li, Huilan,Liu, Chunxia,Wang, Nasi,Huang, Wenlong,Qian, Hai
supporting information, p. 5449 - 5454 (2016/10/22)
The free fatty acid receptor 1 (FFA1/GPR40) is a novel antidiabetic target based on particular mechanism in enhancing glucose-stimulated insulin secretion. Most of reported FFA1 agonists, however, have been suffered from relatively high lipophilicity and
