952235-32-4Relevant academic research and scientific papers
Total syntheses of brominated marine sponge alkaloids
Guinchara, Xavier,Vallee, Yannick,Denis, Jean-Noel
, p. 3761 - 3764 (2007)
Total syntheses of six brominated marine sponge bis(indole) alkaloids of the hamacanthin, spongotine, and topsentin classes are described. Retrosynthetic analysis shows that their structures all include the 1-(6′-bromoindol- 3′-yl)-1,2-diaminoethane unit 13a. This key moiety has been prepared from brominated indolic N-hydroxylamine 5b via synthetic intermediate 8b.
NOVEL BIS-INDOLIC DERIVATIVES, A PROCESS FOR PREPARING THE SAME AND THEIR USES AS A DRUG
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Paragraph 0218; 0223, (2013/03/26)
The present invention relates to novel bis-indolic derivatives, processes for their preparation, and their potential use as new antibacterial drugs.
Novel bis-indolic derivatives, their uses in particular as antibacterials
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Paragraph 0179, (2013/03/26)
The present invention relates to novel bis-indolic derivatives, processes for their preparation, and their potential use as new antibacterial drugs.
BIS-INDOLIC DERIVATIVES, THEIR USES IN PARTICULAR AS ANTIBACTERIALS
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Page/Page column 31, (2013/03/26)
The present invention relates to novel bis-indolic derivatives, processes for their preparation, and their potential use as new antibacterial drugs.
BIS-INDOLIC DERIVATIVES, A PROCESS FOR PREPARING THE SAME AND THEIR USES AS A DRUG
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Page/Page column 40; 42, (2013/03/26)
The present invention relates to novel bis-indolic derivatives, processes for their preparation, and their potential use as new antibacterial drugs.
Synthesis and evaluation of 1-(1H-indol-3-yl)ethanamine derivatives as new antibacterial agents
Burchak, Olga N.,Pihive, Emmanuelle Le,Maigre, Laure,Guinchard, Xavier,Bouhours, Pascale,Jolivalt, Claude,Schneider, Dominique,Maurin, Max,Giglione, Carmela,Meinnel, Thierry,Paris, Jean-Marc,Denis, Jean-No?l
, p. 3204 - 3215 (2011/06/25)
A collection of 3-substituted indole derivatives was prepared using nucleophilic addition of indoles to nitrones. The compounds were then tested for their antibacterial activity against almost thirty bacterial strains representative of common human pathog
