95480-01-6Relevant academic research and scientific papers
A diversity-oriented synthesis of bioactive benzanilides via a regioselective C(sp2)-H hydroxylation strategy
Sun, Yong-Hui,Sun, Tian-Yu,Wu, Yun-Dong,Zhang, Xinhao,Rao, Yu
, p. 2229 - 2238 (2016/03/05)
A diversity-oriented synthesis of bioactive benzanilides via C(sp2)-H hydroxylation has been studied. Different regioselectivity was observed with Ru(ii) and Pd(ii) catalysts. The reaction demonstrates excellent regioselectivity, good tolerance
Relationship between the structure and antimycobacterial activity of substituted salicylanilides
Waisser, Karel,Bures, Otakar,Holy, Pavel,Kunes, Jiri,Oswald, Radek,Jiraskova, Lucie,Pour, Milan,Klimesova, Vera,Kubicova, Lenka,Kaustova, Jarmila
, p. 53 - 71 (2007/10/03)
A series of 143 salicylanilides substituted in positions 4 and 5 and in positions 3′ and 4′ was synthesized. The compounds were evaluated for in vitro antimycobacterial activity against Mycobacterium tuberculosis, Mycobacterium kansasii, and Mycobacterium
BORON TRICHLORIDE CATALYZED ORTHO CARBONYLATION OF PHENOLS: SYNTHESIS OF 2-HYDROXY-ARYL-CARBOXYAMIDES AND -KETONES.
Piccolo, Oreste,Filippini, Lucio,Tinucci, Laura,Valoti, Ermanno,Citterio, Attilio
, p. 885 - 892 (2007/10/02)
In the presence of equimolar quantity of BCl3, phenols 1 react with isocyanates and acyl chlorides to give, usually with good-excellent yields, 2-hydroxy-aryl-carboxy-amides 2 and 2-hydroxy-aryl-ketones 3 respectively.A distinctive behaviour of BCl3 in comparison with other Lewis acids is observed.
