97291-62-8Relevant academic research and scientific papers
Fluoroalkyl-substituted cyclopropane derivatives: Synthesis and physicochemical properties
Grygorenko, Oleksandr O.,Chernykh, Anton V.,Olifir, Oleksandr S.,Kuchkovska, Yuliya O.,Volochnyuk, Dmitriy M.,Yarmolchuk, Vladimir S.
, p. 12692 - 12702 (2020/11/10)
A series of all 12 cis- and trans-cyclopropanecarboxylic acids and cyclopropylamines bearing CH2F, CHF2, and CF3 substituents were synthesized by different methods on a multigram scale. Dissociation constants (pKa) and log P values were measured for the o
BENZOFURAN DERIVATIVES AND THEIR USE AS BROMODOMAIN INHIBITORS
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Page/Page column 57, (2019/04/27)
The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.
2,3-DIHYDROBENZOFURANS AS BOROMODOMAIN INHIBITORS
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Page/Page column 57, (2019/04/27)
The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.
PYRIDINONE DICARBOXAMIDE FOR USE AS BROMODOMAIN INHIBITORS
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Page/Page column 77, (2017/03/21)
The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.
PYRIDINE DICARBOXAMIDE DERIVATIVES AS BROMODOMAIN INHIBITORS
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Page/Page column 38, (2017/12/29)
The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.
