99314-92-8Relevant articles and documents
HIV INTEGRASE INHIBITORS
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Page/Page column 18, (2009/09/08)
Pyridopyrimidine carboxamide compounds of Formula I are inhibitors of HIV integrase and inhibitors of HIV replication: wherein R1, R2, R3, R4, R5 and R6 are defined herein. The compounds ar
3-Hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylates-fast access to a heterocyclic scaffold for HIV-1 integrase inhibitors
Kinzel, Olaf D.,Ball, Richard G.,Donghi, Monica,Maguire, Courtney K.,Muraglia, Ester,Pesci, Silvia,Rowley, Michael,Summa, Vincenzo
scheme or table, p. 6556 - 6558 (2009/04/05)
An efficient and reliable synthesis of the heterocyclic scaffold methyl-3-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylate is described. The scope of the synthesis regarding the introduction of substituents on the pyrido-fused ring is explored.
A new route to N2- and N3-substituted-2,3-diaminopyridines. Synthesis of 1- and 3-alkoxycarbonyl-v-triazolo[4,5-b]pyridines
Zecchini,Torrini,Paradisi
, p. 313 - 318 (2007/10/02)
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