USD $5.00-10.00 / Gram
USD $1.00-10.00 / Kilogram
USD $5.00-10.00 / Gram
USD $1.00-10.00 / Kilogram
USD $5.00-10.00 / Gram
USD $2.00-10.00 / Kilogram
USD $2.00-10.00 / Kilogram
USD $5.00-10.00 / Gram
USD $8.20-8.80 / Kilogram
loxo-101 is a potent, atp-competitive trk inhibitor with ic50s in low nanomolar range for inhibition of all trk family members in binding and cellular assays, with 100-fold selectivity over other kinases, with 2 to 20 nm cellular potency against the trka, trkb, and trkc kinases.
product name: loxo-101
alternate name 3s)-n-[5-[(2r)-2-(2,5-difluorophenyl)-1-pyrrolidinyl]pyrazolo[1,5-a]pyrimidin-3-yl]-3-hydroxy-1-pyrrolidinecarboxamide; arry 470; larotrectinib
appearance: crystalline solid
cas no.: 1223403-58-4
molecular formula: c21h22f2n6o2
molecular weight: 428.44
purity: ≥99%
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