1372799-87-5Relevant articles and documents
Synthesis and evaluation of analogues of estrone-3-O-sulfamate as potent steroid sulfatase inhibitors
Lawrence Woo,Leblond, Bertrand,Purohit, Atul,Potter, Barry V.L.
, p. 2506 - 2519 (2012)
Estrone sulfamate (EMATE) is a potent irreversible inhibitor of steroid sulfatase (STS). In order to further expand SAR, the compound was substituted at the 2- and/or 4-positions and its 17-carbonyl group was also removed. The following general order of p