152171-13-6Relevant articles and documents
Asymmetric Organocatalytic Synthesis of Bisindoles – Scope and Derivatizations
Retich, Christina,Br?se, Stefan
, p. 60 - 77 (2018/01/17)
Starting from 3-vinylindoles and glyoxolate imines, we created a library of diverse 4,6-bis(1H-indole-3-yl)piperidine 2-carboxylates by using 10 mol-% of a chiral phosphoric acid. Utilising electron-withdrawing groups on the starting material during the r
SN2′ boron-mediated Mitsunobu reactions - A new one-pot three-component synthesis of substituted enamides and enol benzoates
Berree, Fabienne,Gernigon, Nicolas,Hercouet, Alain,Chia, Hui Lin,Carboni, Bertrand
supporting information; experimental part, p. 329 - 333 (2009/07/04)
The conversion of (3-hydroxy-1-propen-1-yl)boronates to substituted enamides and enol benzoates is readily achieved in a one-pot procedure consisting of a regiocontrolled Mitsunobu reaction with convenient nucleophiles, followed by allylboration of aldehydes. Wiley-VCH Verlag GmbH & Co. KGaA, 2009.
Rhodium-catalyzed hydroformylation of 2-vinyl- and 3-vinyl-1-tosylpyrroles as a convenient synthetic route to the corresponding 2-(1-tosylpyrrolyl)propanals and derivatives
Settambolo, Roberta,Caiazzo, Aldo,Lazzaroni, Raffaello
, p. 4111 - 4120 (2007/10/03)
2-(1-Tosylpyrrolyl)propanals 2a-b were conveniently prepared (70% yield) via rhodium-catalyzed hydroformylation of the corresponding 2-vinyl- and 3-vinyl-1-tosylpyrroles 1a-b and successfully transformed into some new derivatives (50-90% yield).