191352-29-1Relevant articles and documents
BENZODICYCLOALKANE DERIVATIVE, PREPARATION METHOD AND USE THEREOF
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Paragraph 0348; 0351, (2019/06/19)
It is provided herein a benzobicycloalkane derivative, and a preparation method and use thereof. In particular, it is provided herein a compound of Formula (I), or a pharmaceutically acceptable salt, stereoisomer or solvate thereof, a preparation method, and a use thereof in preparation of drugs for treating pain.
GLUCURONIDE PRODRUGS OF JANUS KINASE INHIBITORS
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Paragraph 0299; 0305; 0306, (2018/12/11)
The invention relates to glucuronide prodrug compounds of Janus kinase (JAK) inhibitors having formula I: where W1, R1 and A1 are as defined. The invention also relates to pharmaceutical compositions comprising such compounds; methods of using such compounds to treat gastrointestinal inflammatory diseases; and processes and intermediates for preparing such compounds.