- Efficient Synthesis of Substituted Morpholine Derivatives via an Indium(III)-catalyzed Reductive Etherification Reaction
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An efficient synthesis of morpholine derivatives has been developed using indium(III)-catalyzed intramolecular reductive etherification reaction. This method allows the construction of various 2-substituted, and 2,3-, 2,5-, 2,6-disubstituted morpholines with good to excellent yields and high diastereoselectivity. In addition, this method demonstrates good compatibility with a broad range of functional groups.
- Fu, Lei,Liu, Haixia,Liu, Yafei,Shen, Hong,Wang, Di,Zhu, Wei
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supporting information
p. 709 - 712
(2020/07/02)
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