Diclofenac derivatives with insulin-sensitizing activity
A series of diclofenac derivatives were synthesized. The insulin-sensitizing activity of 28 new compounds was evaluated in 3T3-L1 cells. The compounds 10a and 10f exhibited similar insulin-sensitizing activity with positive drug rosiglitazone.
Wang, Jian Ta,Wang, Ying,Zhang, Ji Quan,Cui, Xing,Zhang, Yi,Zhu, Gao Feng,Tang, Lei
p. 409 - 412
(2012/01/06)
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