The design and synthesis of a novel series of indole derived selective ETA antagonists
Conformational constraint has been used as the key design element in the identification of a series of potent and selective ETA antagonists. The most potent antagonist, 32, (ETA IC50 = 0.55 nM) is 722-fold selective over t
Rawson, David J.,Dack, Kevin N.,Dickinson, Roger P.,James, Kim
p. 125 - 128
(2007/10/03)
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