cas 345915-64-2, 4-(IODO-PHENYL)-METHANE SULFONYL CHLORIDE

Articles about 345915-64-2Total 3 be found

Synthesis and evaluation of peptidic thrombin inhibitors bearing acid-stable sulfotyrosine analogues
Tyrosine sulfation is an important post-translational modification of peptides and proteins which underpins and modulates many protein-protein interactions. In order to overcome the inherent instability of the native modification, we report the synthesis of two sulfonate analogues and their incorporation into two thrombin-inhibiting sulfopeptides. The effective mimicry of these sulfonate analogues for native sulfotyrosine was validated in the context of their thrombin inhibitory activity and binding mode, as determined by X-ray crystallography.
Agten, Stijn M.,Calisto, Bárbara M.,Dowman, Luke J.,Payne, Richard J.,Pereira, Pedro José Barbosa,Ripoll-Rozada, Jorge
supporting information
p. 10923 - 10926
(2021/10/22)

Synthesis of α-fluorosulfonamides by electrophilic fluorination
(Chemical Equation Presented) α-Fluorosulfonamides were prepared by electrophilic fluorination of tertiary sulfonamides using N- fluorobenzenesulfonimide as fluorinating agent and utilizing the dimethoxybenzyl group (DMB) as a new sulfonamide protecting g
Hill, Bryan,Liu, Yong,Taylor, Scott D.
p. 4285 - 4288
(2007/10/03)

Synthesis of Protected L-4-[Sulfono(difluoromethyl)]phenylalanine and Its Incorporation into a Peptide
matrix presented A protected form of L-4-[sulfono(difluoromethyl)]phenylalanine (F2Smp), a novel non-hydrolyzable phospho- and sulfotyrosine mimetic, was synthesized via electrophilic fluorination of a benzylic sulfonate followed by a Pd-cataly
Liu, Shifeng,Dockendorff, Chris,Taylor, Scott D.
p. 1571 - 1574
(2007/10/03)