503470-23-3Relevant articles and documents
ISOXAZOLINE DERIVATIVES AS PESTICIDES
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Page/Page column 71-72, (2021/06/26)
The present invention provides compounds of formula (I): which are useful for long-lasting treatment and control of pests, for example fleas and ticks, in companion animals and livestock, and pharmaceutical compositions and methods of using the same.
Method for preparing oxazoline insecticide flunia intermediate
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, (2021/04/28)
The invention discloses a method for preparing an oxazoline insecticide fluralan intermediate, the intermediate is 4-formyl-2-methyl benzoic acid, the synthesis route is a certain embodiment of the invention, the limitation that the reaction operation is shortened as much as possible in the prior art is broken through, hydrolysis operation is carried out firstly, and then oxidation reaction is carried out. and the method for preparing oxazoline insecticide flunia intermediate is mild in reaction condition, easy to realize industrially, safe and environment-friendly, and can obtain the low-impurity oxazoline insecticide flunixin intermediate.
Fluorine thramine intermediate and method for preparing flumbine by using same
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Paragraph 0107-0109, (2021/12/07)
The invention discloses a fluororesonide intermediate and a method for preparing the same, and a fluororesonide intermediate -5. Routes include the use of m-xylene as starting materials, halogenation. Oxidation reaction The intermediate -5 is further obtained by hydroximation, cyanolation, hydrolysis reaction or cyanation, oximation, and hydrolysis reaction. As some examples of the present invention, synthetic routes were increased 2 steps from 5 steps in the prior art, but surprisingly high overall yields were obtained and the purity of intermediate -5 was significantly increased. , The starting material of the intermediate -5 is prepared from high 4 - bromo -2 - methylbenzoic acid to low-priced m-xylene, so that the cost of the intermediate -5 is greatly reduced. , The reaction condition is mild, the synthesis difficulty is low, and the environment is more environmentally friendly.
MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS
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Paragraph 00883, (2017/08/01)
Provided herein are antibacterial compounds, wherein the compounds in some embodiments have broad spectrum bioactivity. In various embodiments, the compounds act by inhibition of bacterial type 1 signal peptidase (SpsB), an essential protein in bacteria. Pharmaceutical compositions and methods for treatment using the compounds described herein are also provided.
Pesticidal compositions and processes related thereto
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Page/Page column 50, (2016/01/09)
This document discloses molecules having the following formula (“Formula One”): and processes associated therewith.
PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO
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Paragraph 0240, (2015/12/30)
This disclosure relates to the field of molecules having pesticidal utility against pests in Phyla Nematoda, Arthropoda, and/or Mollusca, processes to produce such molecules and intermediates used in such processes, compositions containing such molecules, and processes of using such molecules against such pests. These molecules may be used, for example, as nematicides, acaricides, insecticides, miticides, and/or molluscicides. This document discloses molecules having the following formula (“Formula One”).
PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO
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Page/Page column, (2014/06/25)
This document discloses molecules having the following formula (“Formula One”): and processes associated therewith.
PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO
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Page/Page column 50, (2014/07/08)
This document discloses molecules having the following formula ("Formula One"): and processes associated therewith.
PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO
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Paragraph 0219, (2014/06/25)
This document discloses molecules having the following formula (“Formula One”): and processes associated therewith.
PESTICIDAL COMPOSITIONS AND PROCESSES RELATED THERETO
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Paragraph 0295, (2014/06/25)
This document discloses molecules having the following formula (“Formula One”): and processes associated therewith.