- Pharmacologically active pyrrolodiazepines
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Compounds of the following formula STR1 wherein R is hydrogen, methyl, ethyl, propyl, isopropyl, butyl, isobutyl, sec.-butyl or tert.-butyl; R1 is hydrogen, methyl, ethyl or phenyl; R2 is hydrogen, methyl, ethyl, propyl, isopropyl, butyl, isobutyl, sec.-butyl or tert.-butyl; R3 is hydrogen, methoxy, trifluoromethyl, chloro, bromo or fluoro; and R4 is methyl. The new compounds are useful as CNS depressants, anticonvulsants, anti-inflammatories and inhibitors of the enzymes which promote the synthesis of prostaglandins.
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