- 1,3-Oxazole-isoniazid hybrids: Synthesis, antitubercular activity, and their docking studies
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A series of novel N′-([2-aryl-5-methyl-1,3-oxazole-4-yl]methylene)isonicotino/nicotino hydrazides 10a-l were prepared by the condensation reaction of 2-aryl-5-methyl-1,3-oxazole-4-carbaldehydes 8a-f with the corresponding isonicotino/nicotino hydrazides 9
- Katariya, Kanubhai D.,Shah, Shailesh R.
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- The synthesis and activity of oxazole and thiazole analogues of urocanic acid
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Direct exposure of human skin to sunlight leads to suppression of the immune system, believed to be mediated by urocanic acid. The synthesis of oxazole and thiazole analogues of urocanic acid is reported, as is their effect on biological markers of the hu
- Millan, David S.,Prager, Rolf H.,Brand, Catherine,Hart, Prue H.
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p. 811 - 816
(2007/10/03)
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- Thiazolidinedione derivatives as hypoglycemic agents
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Hypoglycemic thiazolidine-2,4-dione derivatives of the formula STR1 wherein the dotted line represents a bond or no bond; V is --CH=CH--, --N=CH--, --CH=N--, S, O or NR; W is S, SO, SO2, SO2 NR1, NR1 SO2/s
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- Novel Thiazolidine-2,4-diones as Potent Euglycemic Agents
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A new series of thiazolidine-2,4-diones was obtained by replacing the ether function of englitazone with various functional groups, i.e., a ketone, alcohol, or olefin moiety.These compounds lower blood glucose levels in the genetically obese and insulin-r
- Hulin, Bernard,Clark, David A.,Goldstein, Steven W.,McDermott, Ruth E.,Dambek, Paul J.,et al.
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p. 1853 - 1864
(2007/10/02)
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- Thiazolidinedione derivatives as hypoglycemic agents
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Hypoglycemic thiazolidine-2,4-dione derivatives of the formula wherein the dotted line represents a bond or no bond;, V is -CH=CH-, -N=CH-, -CH=N-, S, O or NR;, W is S, SO, SO2, SO2NR1, NR1SO2, CONR1 or NR1CO;, X is S, O,
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