- Alkylamino derivatives of 4-aminomethylpyridine as inhibitors of copper-containing amine oxidases
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The first substratelike, reversible inhibitors of different copper amine oxidases (CAOs) with IC50 (M) as low as 2.0 × 10-8 corresponding to derivatives of 4-aminomethylpyridine with alkoxy (1a-d), alkylthio (2a,b), and alkylamino (3
- Bertini, Vincenzo,Buffoni, Franca,Ignesti, Giovanni,Picci, Nevio,Trombino, Sonia,Iemma, Francesca,Alfei, Silvana,Pocci, Marco,Lucchesini, Francesco,De Munno, Angela
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p. 664 - 670
(2007/10/03)
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- A Versatile Synthesis of 3H-1(H),4(H)-Benzodiazepin-2,5-diones
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Reaction of isatoic anhydrides (1) and α-amino acids (2) in glacial acetic acid under reflux gave 3H-1(H),4(H)-benzodiazepin-2,5-diones (3) in good yields.These compounds have been characterised by UV, IR, mass, PMR and 13C-NMR spectra.
- Mohiuddin, G.,Reddy, P. S. N.,Ahmed, Khalil,Ratnam, C. V.
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p. 905 - 907
(2007/10/02)
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