- Synthesis of 2-[(4-amino or 2,4-diaminophenyl)sulfonyl] derivatives of benzimidazole, benzothiazole and 6-methyluracil as potential antimicrobial agents
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The synthesis of 2-[(4-aminophenyl)sulfonyl] derivatives of benzimidazole 1 benzothiazole 2 and 6-methyluracil 5 has been accomplished via KMnO4-oxidation of the corresponding 2-(4-nitrophenyl)thio derivatives to the sulfones followed by dissol
- Ghoneim,Essawi,Mohamed,Kamal,Abd El-Megid
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p. 904 - 911
(2007/10/03)
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- Synthesis of 2-Arylthio- and 2-Arylsulphono-benzimidazoles and of 2,4-Dinitro-12(H)-oxo-benzimidazobenzothiazine as Anthelmintic and Antimicrobial Agents
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The synthesis and biological activity of a series of 2-arylthiobenzimidazoles (6, 7, 9, 19, 20 and 24), 2-arylsulphonobenzimidazoles (10-18 and 21-23) and 2,4-dinitro-12(H)-oxobenzimidazobenzothiazine (26) are described.None of the compounds shows significant anthelmintic activity while some of the compounds exhibit growth inhibitory activity against different strains of bacteria and fungi.
- Rao, K. V. B.,Charles, E. S.,Sharma, Satyavan
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p. 575 - 578
(2007/10/02)
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