- HETEROCYCLIC AMINO BERBAMINE DERIVATIVES, PREPARATION METHOD AND USE THEREOF
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The present invention relates to a novel berbamine derivative of formula I or a pharmaceutically acceptable salt thereof, a process for preparation of the same, a pharmaceutical composition comprising said compound and its use in manufacture of an antitumor medicament.
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Paragraph 0095; 0097
(2013/07/25)
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- Tandem photoarylation-photoisomerization of halothiazoles: Synthesis, photophysical and singlet oxygen activation properties of ethyl 2-arylthiazole-5-carboxylates
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The photochemical reaction between ethyl 2-chlorothiazole5-carboxylate and benzene gave no product. In contrast, the reaction with ethyl 2-iodothiazole-5-carboxylate gave ethyl 3-phenylisothiazole-4-carboxylate. The same behaviour was observed if the reac
- Amati, Mario,Belviso, Sandra,D'Auria, Maurizio,Lelj, Francesco,Racioppi, Rocco,Viggiani, Licia
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experimental part
p. 3416 - 3427
(2010/08/20)
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- OPIOID RECEPTOR ANTAGONISTS
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A compound of the formula I: (I) wherein the variables are as described herein, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixture thereof, formulations and methods of use thereof are disclosed.
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Page 26-27; 47
(2010/02/08)
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- Angiotensin II receptor antagonists
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Compounds are disclosed having the formula: STR1 wherein the substituents are defined herein. The compounds of the invention are angiotensin II receptor antagonists.
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- SYNTHESIS OF HALOGENATED THIAZOLE DERIVATIVES OF OLIGO-N-METHYLPYRROLECARBOXAMIDE AND THEIR PHOTOCHEMICAL DNA CLEAVING ACTIVITIES
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Synthesis of various halogenated thiazole derivatives of oligo-N-methylpyrrolecarboxamide and their DNA cleaving activities under UV-A irradiation were described.
- Sakai, Yasuhiro,Matsumoto, Toyomi,Tanaka, Akie,Shibuya, Masayuki
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p. 565 - 573
(2007/10/02)
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