Potent oxindole based human β3 adrenergic receptor agonists
The synthesis and biological evaluation of a series of oxindole β3 adrenergic receptor agonists is described. A modulation of rat atrial tachycardia was observed with substitution at the 3-position of the oxindole moiety.
Stevens, F. Craig,Bloomquist, William E.,Borel, Anthony G.,Cohen, Marlene L.,Droste, Christine A.,Heiman, Mark L.,Kriauciunas, Aidas,Sall, Daniel J.,Tinsley, Frank C.,Jesudason, Cynthia D.
p. 6270 - 6273
(2008/09/17)
Dehydrogenation of Indolines to Indoles via Azasulphonium Salts or N-Chloramines
The dehydrogenation of indolines to indoles without using mineral oxidising reagents is described.The conversion was achieved via either azasulphonium salts or N-chloramines, the former route involving milder conditions but a more complex procedure.
Kawase, Masami,Miyake, Yuko,Kikugawa, Yasuo
p. 1401 - 1404
(2007/10/02)
More Articles about upstream products of 93831-00-6