TRPV1 modulators: Structure-activity relationships using a rational combinatorial approach

DOI: 10.1016/j.bmcl.2011.04.141

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 3541 - 3545 (2011)

Update date:2022-09-26

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Authors:

Zaccaro, Laura

Garcia-Lopez, M. Teresa

Gonzalez-Muniz, Rosario

Garcia-Martinez, Carolina

Ferrer-Montiel, Antonio

Albericio, Fernando

Royo, Miriam

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Article abstract of DOI:10.1016/j.bmcl.2011.04.141

A discrete library of linear and hydantoin-containing dipeptide derivatives, based on the Lys-Trp(Nps) scaffold, was prepared by solid-phase synthesis. SAR studies indicated that potency for TRPV1 blockade and selectivity towards NMDA is mainly dictated b

Full text of DOI:10.1016/j.bmcl.2011.04.141

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