Peptide modification by introduction of α-trifluoromethyl α-amino acids via 4-trifluoromethyl-1,3-oxazolidin-2,5-diones

Article abstract of DOI:10.1016/0040-4039(92)88047-9

α-Trifluoromethyl substituted α-amino acids can be introduced into the N-terminal position of peptides on carboxyl group activation via Leuchs anhydrides.