Addition of molecular fluorine to azlactones: General synthetic method of erythro-β-fluorinated α-amino acids

DOI: 10.1248/cpb.43.760

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 760 - 765 (1995)

Update date:2022-08-04

Topics:

Authors:

Kaneko Kaneko

Chiba Chiba

Toyota Toyota

Sato Sato

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.43.760

Reaction of molecular fluorine with unsaturated azlactones derived from appropriate aldehydes (or ketones) and benzoylglycine afforded the difluorinated adducts. The reductive amination reaction of the β-fluorinated α-oxoalkanoic acids obtained from the a

Full text of DOI:10.1248/cpb.43.760

NII-Electronic Library Service

Products guided by the article

Product name:4-Fluoro-4-(1-fluoro-1-methyl-ethyl)-2-phenyl-4H-oxazol-5-one

Cas No:171078-05-0

R&D Labs maybe for 171078-05-0

HAORUI ENTERPRISES LLC

Contact:(1) 206-3550089

Address:5115 NE 8TH PL, Renton, WA 98059 USA
Nowa pharmaceuticals Co., LTD

Contact:86-512-69362780,69362785

Address:No.69 Weixin Road,Weiting Town,Suzhou Industrial Park
Tianjin Dongchang Fine Chemical Industry Co., Ltd.

Contact:+86-22-29894595

Address:Economic Developing Zone, Ji County, Tianjin, China
Hebei Lead Bio-Chemicals Co., Ltd.

website:http://www.ldbiochem.com

Contact:+86-311-87826503

Address:481, Heping West Road, Shijiazhuang,China
STAR SYNTHESIS CO.,LIMITED

Contact:+(852) 301-98033

Address:Flat C, 23/F, Lucky Plaza, 315-321 Lockhart Road, Wan Chai, Hong Kong

Relevant to this article

A Novel Oxidative Cyclization of 2'-Hydroxychalcones to 4,5-Dialkoxyaurones by Thallium(III) Nitrate

Doi:10.1021/jo00125a041
(1995)
Fluoro organics: synthesis of novel fluorinated 4-oxo-4H-pyrido<3',2':4,5>furo<3,2-d>-1,3-oxazines and their reactions

Doi:10.1016/0022-1139(95)03239-A
(1995)
An unprecedented photochemical Cis to Trans isomerization of dinuclear gold(I) bis(diphenylphosphino)ethylene complexes

Doi:10.1021/ja00142a041
(1995)
Mild Friedel-Crafts Reactions Enable a Robust Synthesis of Roseophilin

Doi:10.1021/acs.orglett.9b01100
(2019)
Activation of carboxylic acids by pyrocarbonates. Application of di-tert-butyl pyrocarbonate as condensing reagent in the synthesis of amides of protected amino acids and peptides

Doi:10.1016/0040-4039(95)01412-B
(1995)
ACETALS OF LACTAMS AND AMIDES OF ACIDS. COMMUNICATION 78. SYNTHESIS AND BIOLOGICAL ACTIVITY OF 7,8-POLYMETHYLENEPURINE DERIVATIVES

Doi:10.1007/BF02226520
(1995)

Article Doi