Addition of molecular fluorine to azlactones: General synthetic method of erythro-β-fluorinated α-amino acids

DOI: 10.1248/cpb.43.760

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 760 - 765 (1995)

Update date:2022-08-04

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Authors:

Kaneko Kaneko

Chiba Chiba

Toyota Toyota

Sato Sato

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Article abstract of DOI:10.1248/cpb.43.760

Reaction of molecular fluorine with unsaturated azlactones derived from appropriate aldehydes (or ketones) and benzoylglycine afforded the difluorinated adducts. The reductive amination reaction of the β-fluorinated α-oxoalkanoic acids obtained from the a

Full text of DOI:10.1248/cpb.43.760

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