Enantioselective Friedel-Crafts alkylation of indole derivatives catalyzed by new Yb(OTf)3-pyridylalkylamine complexes as chiral Lewis acids

DOI: 10.1039/c0ob00461h

Source and publish data:

Organic and Biomolecular Chemistry p. 497 - 503 (2011)

Update date:2022-07-31

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Authors:

Grach, Guillaume

Dinut, Aurelia

Marque, Sylvain

Marrot, Jerome

Gil, Richard

Prim, Damien

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Article abstract of DOI:10.1039/c0ob00461h

New Yb(OTf)₃-pyridylalkylamine complexes have been employed as chiral Lewis acids in the enantioselective Friedel-Crafts alkylation of indole derivatives with trifluoropyruvates. The influence of the substituents as well as the configuration of

Full text of DOI:10.1039/c0ob00461h

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