Journal of Medicinal Chemistry p. 12542 - 12573 (2020)
Update date:2022-08-15
Topics:
Fairhurst, Robin A.
Knoepfel, Thomas
Buschmann, Nicole
Leblanc, Catherine
Mah, Robert
Todorov, Milen
Nimsgern, Pierre
Ripoche, Sebastien
Niklaus, Michel
Warin, Nicolas
Luu, Van Huy
Madoerin, Mario
Wirth, Jasmin
Graus-Porta, Diana
Weiss, Andreas
Kiffe, Michael
Wartmann, Markus
Kinyamu-Akunda, Jacqueline
Sterker, Dario
Stamm, Christelle
Adler, Flavia
Buhles, Alexandra
Schadt, Heiko
Couttet, Philippe
Blank, Jutta
Galuba, Inga
Trappe, J?rg
Voshol, Johannes
Ostermann, Nils
Zou, Chao
Berghausen, J?rg
Del Rio Espinola, Alberto
Jahnke, Wolfgang
Furet, Pascal
FGF19 signaling through the FGFR4/β-klotho receptor complex has been shown to be a key driver of growth and survival in a subset of hepatocellular carcinomas, making selective FGFR4 inhibition an attractive treatment opportunity. A kinome-wide sequence al
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