Bioorganic and Medicinal Chemistry Letters p. 2599 - 2602 (1999)
Update date:2022-08-29
Topics:
Lavergne, Olivier
Harnett, Jeremiah
Rolland, Alain
Lanco, Christophe
Lesueur-Ginot, Laurence
Demarquay, Daniele
Huchet, Marion
Coulomb, Helene
Bigg, Dennis C. H.
BN 80927, a novel homocamptothecin derivative, inhibits both topoisomerase I and topoisomerase II mediated DNA relaxation and shows pronounced cytotoxicity against HT29, SKOV-3, DU145 and MCF7 human tumor cell lines.
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(2013)