Bioorganic and Medicinal Chemistry Letters p. 905 - 911 (2019)
Update date:2022-08-16
Topics:
Zhang, Birong
Kiefer, James R.
Blake, Robert A.
Chang, Jae H.
Hartman, Steven
Ingalla, Ellen Rei
Kleinheinz, Tracy
Mody, Vidhi
Nannini, Michelle
Ortwine, Daniel F.
Ran, Yingqing
Sambrone, Amy
Sampath, Deepak
Vinogradova, Maia
Zhong, Yu
Nwachukwu, Jerome C.
Nettles, Kendall W.
Lai, Tommy
Liao, Jiangpeng
Zheng, Xiaoping
Chen, Hai
Wang, Xiaojing
Liang, Jun
Despite tremendous progress made in the understanding of the ERα signaling pathway and the approval of many therapeutic agents, ER+ breast cancer continues to be a leading cause of cancer death in women. We set out to discover compounds with a dual mechan
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