Z-ASP(OSU)-OBZL

Base Information

• Chemical Name: Z-ASP(OSU)-OBZL
• CAS No.: 108325-86-6
• Molecular Formula: C23H22 N2 O8
• Molecular Weight: 454.43
• Mol file: 108325-86-6.mol

Synonyms:Z-ASP(OSU)-OBZL;Z-ASPARTIC ACID(OSU)-OBZL;Z-L-ASPARTIC ACID BETA-N-HYDROXYSUCCINIMIDE ESTER ALPHA-BENZYL ESTER

Chemical Property of Z-ASP(OSU)-OBZL

Chemical Property:

• PSA: 128.31000
• LogP: 2.35090
• Storage Temp.: -15°C

Purity/Quality:

99% ^*data from raw suppliers

Z-ASP(OSU)-OBZL ^*data from reagent suppliers

Safty Information:

• Pictogram(s):  
• Hazard Codes: 

MSDS Files:

SDS file from LookChem

Useful:

Technology Process of Z-ASP(OSU)-OBZL

There total 1 articles about Z-ASP(OSU)-OBZL which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

1-hydroxy-pyrrolidine-2,5-dione (6066-82-6) + Z-Asp-OBn (4779-31-1) → 1-benzyl N-benzyloxycarbonyl-4-(N-succinimido)-L-aspartate (108325-86-6)

Guidance literature:

With dicyclohexyl-carbodiimide; In 1,2-dimethoxyethane; Yield given; -10 deg C, 1 h; -5 deg C, 18 h;

DOI:10.1007/BF00954837

Reference yield: 82.0%

Tyr(tBu) (16874-12-7,87553-74-0) + 1-benzyl N-benzyloxycarbonyl-4-(N-succinimido)-L-aspartate (108325-86-6) → (S)-2-Benzyloxycarbonylamino-N-[(S)-1-tert-butoxycarbonyl-2-(4-hydroxy-phenyl)-ethyl]-succinamic acid benzyl ester (178271-91-5)

Guidance literature:

With triethylamine; In dichloromethane; water; N,N-dimethyl-formamide; 1.) 0 deg C, 1 h, 2.) RT, 15 h;

DOI:10.1021/ja952265x

Reference yield: 37.0%

N,N'-diacetylchitobiosamine (102039-77-0) + 1-benzyl N-benzyloxycarbonyl-4-(N-succinimido)-L-aspartate (108325-86-6) → 2-acetamido-4-O-(2-acetamido-2-deoxy-β-D-glucopyranosyl)-1-N-(1-benzyloxy-N-benzyloxycarbonyl-4-L-aspartyl)-2-deoxy-β-D-glucopyranosylamine

Guidance literature:

In water; N,N-dimethyl-formamide; at 20 ℃; for 16h;

DOI:10.1007/BF00954837

upstream raw materials:

1-hydroxy-pyrrolidine-2,5-dione

Z-Asp-OBn

Downstream raw materials:

(S)-2-Benzyloxycarbonylamino-N-[(S)-1-tert-butoxycarbonyl-2-(4-hydroxy-phenyl)-ethyl]-succinamic acid benzyl ester

(S)-2-Benzyloxycarbonylamino-N-[(S)-1-carboxy-2-(4-hydroxy-phenyl)-ethyl]-succinamic acid benzyl ester

Post a RFQ

Cas No.:

Product Name:

Quantity:

Please select Metric Ton KG G Pound L ML

Email:

Company name:

Valid Period:

Detailed Requirements:

• Sample
• MOQ
• GMP
• FDA
• Price
  FOB CIF CFR EXW
• Urgent purchase

Enter 15 to 2000 letters.Word count: 0 letters

Attach files(File Format: Jpeg, Jpg, Gif, Png, PDF, PPT, Zip, Rar,Word or Excel Maximum File Size: 3MB)

Remove

Submit

1

What can I do for you?
Get Best Price

Get Best Price for 108325-86-6 Z-ASP(OSU)-OBZL

Send

Send

Metric Ton KG G Pound L ML

Send

Send