(2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate

Base Information

Chemical Name:(2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate
CAS No.:1093878-47-7
Molecular Formula:C₂HF₃O₂*C₁₀H₁₂BF₂NO₃
Molecular Weight:357.042
Hs Code.:

Synonyms:(2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate

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Chemical Property of (2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate

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Technology Process of (2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate

There total 2 articles about (2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

: 121-43-7,63156-11-6
Trimethyl borate

: 736991-31-4
4-(3,5-difluorophenyl)morpholine

: 76-05-1
trifluoroacetic acid

: 1093878-47-7
(2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate

Guidance literature:: 4-(3,5-difluorophenyl)morpholine; With n-butyllithium; diisopropylamine; In tetrahydrofuran; at -78 ℃; for 0.5h;

Trimethyl borate; In tetrahydrofuran; at -78 - 20 ℃;

trifluoroacetic acid;

Reference yield:

: 461-96-1
3,5-difluorobromobenzene

: 1093878-47-7
(2,6-difluoro-4-morpholin-4-ylphenyl)boronic acid trifluoroacetate

Guidance literature:: Multi-step reaction with 2 steps

1.1: potassium carbonate; XPhos / tris-(dibenzylideneacetone)dipalladium⁽⁰⁾ / tert-Amyl alcohol / 100 °C / Inert atmosphere

2.1: diisopropylamine; n-butyllithium / tetrahydrofuran / 0.5 h / -78 °C

2.2: -78 - 20 °C

With n-butyllithium; potassium carbonate; diisopropylamine; XPhos; tris-(dibenzylideneacetone)dipalladium⁽⁰⁾; In tetrahydrofuran; tert-Amyl alcohol;