(R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester

Base Information

Chemical Name:(R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester
CAS No.:203639-76-3
Molecular Formula:C₂₄H₂₁IN₂O₄S
Molecular Weight:560.412
Hs Code.:

Synonyms:(R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester

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Chemical Property of (R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester

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Technology Process of (R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester

There total 2 articles about (R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

: 126090-33-3
(R)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionic acid benzyl ester

: 203639-76-3
(R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester

Guidance literature:: Multi-step reaction with 2 steps

1: CH₂Cl₂ / 1 h / Ambient temperature

2: N-methylmorpholine / CH₂Cl₂ / 2 h / Ambient temperature

With 4-methyl-morpholine; In dichloromethane;
DOI:10.1021/jm9707582

Reference yield:

: 98-61-3
p-Iodobenzenesulfonyl chloride

: D-tryptophan benzyl ester trifluoroacetate

: 203639-76-3
(R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester

Guidance literature:: With 4-methyl-morpholine; In dichloromethane; for 2h; Ambient temperature;
DOI:10.1021/jm9707582

Reference yield:

: 203639-76-3
(R)-3-(1H-Indol-3-yl)-2-(4-iodo-benzenesulfonylamino)-propionic acid benzyl ester

: (R)-3-(1H-indol-3-yl)-2-(4'-methoxybiphenyl-4-sulfonylamino)propionic acid

Guidance literature:: Multi-step reaction with 2 steps

1: Pd(PPh₃)4, K₂CO₃ / tetrahydrofuran / 75 °C

2: H₂ / 10percent Pd/C / methanol; ethyl acetate

With tetrakis(triphenylphosphine) palladium⁽⁰⁾; hydrogen; potassium carbonate; palladium on activated charcoal; In tetrahydrofuran; methanol; ethyl acetate;
DOI:10.1021/jm9707582