183609-18-9Relevant articles and documents
Triazole compound and application thereof in agriculture (by machine translation)
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Paragraph 0240-0242; 0244-0246, (2020/02/10)
More specifically, the present invention relates to a; method for, preparing a triazole compound (I) represented by formula (I) or a salt (I) thereof, a salt thereof, and a method, for producing a, triazole compound, a salt thereof, and a method for controlling a, disease by using these compounds, and or compositions in the form of a fungicide and a; fungicide ,R composition thereof. 1 , R2 , Y, n, X, R3 , R4 The, m invention has Het .the meanings as described in the present invention. (by machine translation)
Discovery of 5-phenoxy-1,3-dimethyl-1H-pyrazole-4-carboxamides as potent agonists of TGR5 via sequential combinatorial libraries
Londregan, Allyn T.,Piotrowski, David W.,Futatsugi, Kentaro,Warmus, Joseph S.,Boehm, Markus,Carpino, Philip A.,Chin, Janice E.,Janssen, Ann M.,Roush, Nicole S.,Buxton, Joanne,Hinchey, Terri
, p. 1407 - 1411 (2013/03/14)
Optimization of a high-throughput screening hit led to the discovery of a new series of 5-phenoxy-1,3-dimethyl-1H-pyrazole-4-carboxamides as highly potent agonists of TGR5. This novel chemotype was rapidly developed through iterative combinatorial library synthesis. It was determined that in vitro agonist potency correlated with functional activity data from human peripheral blood monocytes.
Synthesis of C-aryl-N-cyclopropylnitrones
Vukics, Krisztina,Tarkanyi, Gabor,Dravecz, Ferenc,Fischer, Janos
, p. 3419 - 3425 (2007/10/03)
Synthesis of C-aryl-N-cyclopropylnitrones is described. Preparations were performed either by condensation of the appropriate aldehyde with N-cyclopropyl-hydroxylamine, or oxidation of N-substituted N-cyclopropylamines with sodium tungstate/hydrogen perox
