1000183-50-5Relevant academic research and scientific papers
Design, synthesis and biological profiling of aryl piperazine based scaffolds for the management of androgen sensitive prostatic disorders
Gupta, Sonal,Pandey, Deepti,Mandalapu, Dhanaraju,Bala, Veenu,Sharma, Vikas,Shukla, Mahendra,Yadav, Santosh K.,Singh, Nidhi,Jaiswal, Swati,Maikhuri, Jagdamba P.,Lal, Jawahar,Siddiqi, Mohammad I.,Gupta, Gopal,Sharma, Vishnu L.
, p. 2111 - 2121 (2016)
In the quest for novel scaffolds for the management of androgen sensitive prostatic disorders like prostate cancer and benign prostatic hyperplasia, a series of twenty-six aryl/heteroaryl piperazine derivatives have been described. Three compounds, 8a, 8c
3,5-DIAMINOPYRAZOLE KINASE INHIBITORS
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Paragraph 00435, (2013/09/26)
Provided herein are 3,5-diaminopyrazoles, for example, compounds of Formula IA, that are useful for modulating regulated-in-COPD kinase activity, and pharmaceutical compositions thereof. Also provided herein are methods of their use for treating, preventi
TYROSINE KINASE INHIBITORS
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Page/Page column 63-64, (2008/06/13)
The present invention relates to 4-indol-3-yl-N-phenylpyrimidin-2-amine derivatives, that are useful for treating cellular proliferative diseases, for treating disorders associated with MET activity, and for inhibiting the receptor tyrosine kinase MET. Th
