1001333-82-9Relevant academic research and scientific papers
Design and evaluation of novel biphenyl sulfonamide derivatives with potent histamine H3 receptor inverse agonist activity
Covel, Jonathan A.,Santora, Vincent J.,Smith, Jeffrey M.,Hayashi, Rena,Gallardo, Charlemagne,Weinhouse, Michael I.,Ibarra, Jason B.,Schultz, Jeffrey A.,Park, Douglas M.,Estrada, Scott A.,Hofilena, Brian J.,Pulley, Michelle D.,Smith, Brian M.,Ren, Albert,Suarez, Marissa,Frazer, John,Edwards, Jeffrey,Hauser, Erin K.,Lorea, Jodie,Semple, Graeme,Grottick, Andrew J.
, p. 5603 - 5611 (2009)
Antagonism of the histamine-H3 receptor is one tactic being explored to increase wakefulness for the treatment of disorders such as excessive daytime sleepiness (EDS) as well as other sleep or cognitive disorders. Phenethyl-R-2-methylpyrrolidin
Tetrahydroimidazo[1,5-d][1,4]oxazepine compound
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Paragraph 0149; 0150; 0151, (2016/03/14)
A compound represented by formula (I): wherein R is a methyl group or the like, R1 is a fluorine atom or the like, R2 is a hydrogen atom or a fluorine atom, R3 is a hydrogen atom, R4 is an ethyl group or the lik
ARYL SULFONAMIDES USEFUL FOR MODULATION OF THE PROGESTERONE RECEPTOR
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Page/Page column 12, (2008/12/08)
In one embodiment, compounds of the following structure are described, wherein R1 to R7 are described herein. Also provided are methods for preparing these compounds and methods of contraception; treating or preventing fibroids; trea
