1011265-01-2Relevant academic research and scientific papers
Substituted oxazolidinones as novel NPC1L1 ligands for the inhibition of cholesterol absorption
Pfefferkorn, Jeffrey A.,Larsen, Scott D.,Huis, Chad Van,Sorenson, Roderick,Barton, Tom,Winters, Thomas,Auerbach, Bruce,Wu, Chenyan,Wolfram, Thaddeus J.,Cai, Hongliang,Welch, Kathleen,Esmaiel, Nadia,Davis, JoAnn,Bousley, Richard,Olsen, Karl,Mueller, Sandra Bak,Mertz, Thomas
, p. 546 - 553 (2008/09/19)
Cholesterol absorption inhibition (CAI) represents an important treatment option for hypercholesterolemia. Herein, we report the design and evaluation of a series of substituted oxazolidinones as ligands for the Niemann Pick C1 Like 1 (NPC1L1) protein, a
