1011469-69-4Relevant articles and documents
Synthesis and structure-activity relationship studies of tyrosine-based antagonists at the human P2X7 receptor
Lee, Ga Eun,Joshi, Bhalchandra V.,Chen, Wangzhong,Jeong, Lak Shin,Moon, Hyung Ryong,Jacobson, Kenneth A.,Kim, Yong-Chul
, p. 571 - 575 (2008/09/20)
Analogues of the P2X7 receptor antagonist KN-62, modified at the piperazine and arylsulfonyl groups, were synthesized and assayed at the human P2X7 receptor for inhibition of BzATP-induced effects, that is, uptake of a fluorescent dy