1016259-43-0Relevant articles and documents
Synthesis and biological evaluation of α- and β-6-amido derivatives of 17-cyclopropylmethyl-3,14β-dihydroxy-4, 5α- epoxymorphinan: Potential alcohol-cessation agents
Ghirmai, Senait,Azar, Marc R.,Polgar, Wilma E.,Berzetei-Gurske, Ilona,Cashman, John R.
, p. 1913 - 1924 (2008/12/21)
Substituted aryl and aliphatic amide analogues of 6-naltrexamine were synthesized and used to characterize the binding to and functional activity of human μ-, δ-, and κ-opioid receptors. Competition binding assays showed 11-25 and 27-31 bound to the μ (K