1026874-71-4Relevant articles and documents
Synthesis and characterization of non-steroidal ligands for the glucocorticoid receptor: Selective quinoline derivatives with prednisolone-equivalent functional activity
Coghlan,Kym,Elmore,Wang,Luly,Wilcox,Stashko,Lin,Miner,Tyree,Jacobson,Nakane,Lane
, p. 2879 - 2885 (2001)
A novel class of functional ligands for the human glucocorticoid receptor is described. Substituents in the C-10 position of the tetracyclic core are essential for glucocorticoid receptor (GR) selectivity versus other steroid receptors. The C-5 position i