103500-49-8

Basic information

• Product Name: 6β-<2-acetamido>-17-(cyclopropylmethyl)4,5α-epoxy-3,14-dihydroxymorphinan
• Synonyms: 6β-<2-acetamido>-17-(cyclopropylmethyl)4,5α-epoxy-3,14-dihydroxymorphinan
• CAS NO: 103500-49-8
• Molecular Weight: 533.624
• Mol File: 103500-49-8.mol

Chemical Properties

• CAS DataBase Reference: 6β-<2-acetamido>-17-(cyclopropylmethyl)4,5α-epoxy-3,14-dihydroxymorphinan(CAS DataBase Reference)
• NIST Chemistry Reference: 6β-<2-acetamido>-17-(cyclopropylmethyl)4,5α-epoxy-3,14-dihydroxymorphinan(103500-49-8)
• EPA Substance Registry System: 6β-<2-acetamido>-17-(cyclopropylmethyl)4,5α-epoxy-3,14-dihydroxymorphinan(103500-49-8)

Safety Data

• Hazardous Substances Data: 103500-49-8(Hazardous Substances Data)

Upstream product

• 63463-07-0 beta-Naltrexamine dihydrochloride 
• 41445-61-8 C₁₅H₁₉NO₆ 
• 1138-80-3 N-(Benzyloxycarbonyl)glycine 

Relevant articles and documents

Synthesis and Biological Activity of Analogues of β-Chlornaltrexamine and β-Funaltrexamine at Opioid Receptors

β-Chlornaltrexamine and β-funaltrexamine analogues 4-7 with different length "arms" to which an electrophilic moiety is attached were synthesized in an effort to obtain affinity labels that would selectively and irreversibly block specific opioid receptor types and subtypes.One of the compounds, 4, was a potent, irreversible blocker of opioid receptors in the guinea pig ileum and mouse vas deferens preparations.The results of this study suggest that nucleophiles that are remote from the recognition locus are capable of alkylation by reactive electrophiles.