1044265-99-7Relevant academic research and scientific papers
Design and synthesis of benzenesulfonanilides active against methicillin-resistant Staphylococcus aureus and vancomycin-resistant Enterococcus
Namba, Kensuke,Zheng, Xiaoxia,Motoshima, Kazunori,Kobayashi, Hidetomo,Tai, Akihiro,Takahashi, Eizo,Sasaki, Kenji,Okamoto, Keinosuke,Kakuta, Hiroki
, p. 6131 - 6144 (2008/12/21)
Vancomycin is mainly used as an antibacterial agent of last resort, but recently vancomycin-resistant bacterial strains have been emerging. Although new antimicrobials have been developed in order to overcome drug-resistant bacteria, many are structurally
In vitro PAI-1 inhibitory activity of oxalamide derivatives
Jain, Mukul R.,Shetty, Shankar,Chakrabarti, Ganes,Pandya, Vrajesh,Sharma, Ajay,Parmar, Bhavesh,Srivastava, Soma,Raviya, Mehul,Soni, Hitesh,Patel, Pankaj R.
, p. 880 - 884 (2008/09/20)
A number of oxalamide derivatives have been synthesized and evaluated for PAI-1 inhibitory activity. In vitro PAI-1 inhibitory activities of oxalamide derivatives are evaluated by chromogenic assay. Few compounds have shown significant PAI-1 inhibitory activity.
