105776-29-2Relevant academic research and scientific papers
Dimethoxyindoles based thiosemicarbazones as multi-target agents; synthesis, crystal interactions, biological activity and molecular modeling
Bingul, Murat,Boga, Mehmet,Kandemir, Hakan,Koca, Mehmet Serdar,Saglam, Mehmet F.,Sengul, Ibrahim F.,Temel, Mutesir,Zorlu, Yunus,Y?ld?z, Minhal
, (2022/02/03)
Alzheimer's disease (AD) is known as one of the most devastating neurodegenerative disease diagnosed for the old-aged people and cholinesterase inhibitors (ChEI) can be used as an effective palliative treatment for AD. A range of novel monomeric and dimer
First heterogeneous ligand- and salt-free larock indole Synthesis
Batail, Nelly,Bendjeriou, Anissa,Lomberget, Thierry,Barrett, Roland,Dufaud, Veronique,Djakovitch, Laurent
supporting information; experimental part, p. 2055 - 2062 (2009/12/26)
A new ligand- and salt-free procedure using heterogeneous palladium catalysts for the Larock indole and benzofuran synthesis is reported. After optimisation of the reaction conditions, good to high isolated yields have been achieved for a variety of structures. Recycling studies have shown that the palladium catalysts can be readily recovered and reused. Reactions and recovery of the palladium catalysts can be carried out in the presence of air, without any particular precaution.
Synthesis of activated 3-substituted indoles: An optimised one-pot procedure
Pchalek, Karin,Jones, Ashley W.,Wekking, Monique M.T.,Black, David StC.
, p. 77 - 82 (2007/10/03)
3-Substituted-4,6-dimethoxyindoles can be synthesised in a one-pot procedure from 3,5-dimethoxyaniline and 2-haloketones in the presence of lithium bromide and sodium bicarbonate. Graphical Abstract.
Synthesis of Activated 3-Arylindoles
Black, David St. C.,Bowyer, Michael C.,Bowyer, Paul K.,Ivory, Andrew J.,Kim, Mihyong,et al.
, p. 1741 - 1750 (2007/10/02)
A wide range of substituted 3-aryl-4,6-dimethoxyindoles (6) has been synthesized from the related α-anilinoacetophenones (5), in which the nitrogen atom is protected by a trifluoroacetyl or acetyl group.This method has led to the synthesis of a 3,7'-biindolyl (12).
Synthesis of 4,6-Dimethoxyindoles
Black, David St.C.,Kumar, Naresh,Wong, Laurence C. H.
, p. 15 - 20 (2007/10/02)
Syntheses are described for nine new 4,6-dimethoxyindoles, incorporating phenyl, pyridin-2-yl, methoxycarbonyl, carboxy and methyl groups in the 2- and/or 3-positions.
