1060749-17-8Relevant articles and documents
Anxiolytic-like effects of N,N-dialkyl-2-phenylindol-3-ylglyoxylamides by modulation of translocator protein promoting neurosteroid biosynthesis
Da Settimo, Federico,Simorini, Francesca,Taliani, Sabrina,La Motta, Concettina,Marini, Anna Maria,Salerno, Silvia,Bellandi, Marusca,Novellino, Ettore,Greco, Giovanni,Cosimelli, Barbara,Da Pozzo, Eleonora,Costa, Barbara,Simola, Nicola,Morelli, Micaela,Martini, Claudia
supporting information; experimental part, p. 5798 - 5806 (2009/08/07)
Novel N,N-disubstituted indol-3-ylglyoxylamides (1-56), bearing different combinations of substituents R1-R5, were synthesized and evaluated as ligands of the translocator protein (TSPO), the 18 kDa protein representing the minimal f