1082208-29-4Relevant academic research and scientific papers
Refining the structure?activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms
Magalh?es, Joana,Franko, Nina,Annunziato, Giannamaria,Pieroni, Marco,Benoni, Roberto,Nikitjuka, Anna,Mozzarelli, Andrea,Bettati, Stefano,Karawajczyk, Anna,Jirgensons, Aigars,Campanini, Barbara,Costantino, Gabriele
, p. 31 - 43 (2019)
The lack of efficacy of current antibacterials to treat multidrug resistant bacteria poses a life-threatening alarm. In order to develop enhancers of the antibacterial activity, we carried out a medicinal chemistry campaign aiming to develop inhibitors of
Dramatically accelerated addition under solvent-free conditions: An efficient synthesis of (E)-1,2,4-triazole-substituted alkenes from Baylis-Hillman acetates
Zhong, Weihui,Zhao, Yongzhi,Guo, Baoming,Wu, Peng,Su, Weike
, p. 3291 - 3302 (2008/12/22)
The addition of 1,2,4-triazole to Baylis-Hillman acetates mediated by Et3N was dramatically accelerated under solvent-free conditions to afford (E)-1,2,4-triazole-substituted alkenes 3 with excellent yields. Copyright Taylor & Francis Group, LLC.
