108279-24-9Relevant academic research and scientific papers
ANALOGUES OF THE CHOLECYSTOKININ C-TERMINAL TETRRAPEPTIDE
Hlavacek, Jan,Marcova, Renata,Maletinska, Lenka,Slaninova, Jirina
, p. 2511 - 2522 (2007/10/02)
Substituted phenylethyl amides and phenylethyl esters Va - Vj derived from the carboxyterminal tetrapeptide part of the cholecystokinin were synthesized and their biological properties assayed.In the original CCK tetrapeptide structure Trp-Met-Asp-Phe-NH2
Development of a Small RGD Peptide Fibrinogen Receptor Antagonist with Potent Antiaggregatory Activity in Vitro
Samanen, J.,Ali, F.,Romoff, T.,Calvo, R.,Sorenson, E.,et al.
, p. 3114 - 3125 (2007/10/02)
The development of potent antithrombotic agents from the fibrinogen platelet receptor binding sequences Fg-α 572-575 -Arg-Gly-Asp-Ser- and Fg-γ 400-411 -HHLGGAKQAGDV, believed to be a cryptic RGD-type sequence, is described.The tetrapeptide Ac-RGDS-NH2 it
Synthesis of gastrin antagonists, analogues of the C-terminal tetrapeptide of gastrin, by introduction of a β-homo residue
Rodriguez,Fulcrand,Laur,Aumelas,Bali,Martinez
, p. 522 - 528 (2007/10/02)
A series of analogues of Boc-Trp-Leu-Asp-Phe-NH2, a potent gastrin agonist, were synthesized by introducing a β-homo residue in the sequence. These compounds were tested in vivo on acid secretion, in the anesthetized rat, and for their ability
